Catalog No. Size 价格库存数量
S2242-2 Solid 2 mg ¥90
S2242-10 Solid 10 mg ¥270


Falnidamol, also known as BIBX 1382, is a pyrimido-pyrimidine with antitumor activity. BIBX 1382 inhibits the intracellular tyrosine kinase domain of the Epidermal Growth Factor Receptor (EGFR) thus specifically reversing the aberrant enzymatic activity from overexpressed and constitutively activated EGFR, and subsequently inhibiting cell proliferation and inducing cell differentiation. Check for active clinical trials or closed clinical trials using this agent.

Product information

CAS Number: 196612-93-8

Molecular Weight: 387.84

Formula: C18H19ClFN7

Chemical Name: N8-(3-chloro-4-fluorophenyl)-N2-(1-methylpiperidin-4-yl)-[1,3]diazino[5,4-d]pyrimidine-2,8-diamine

Smiles: CN1CCC(CC1)NC1=NC2=C(NC3=CC(Cl)=C(F)C=C3)N=CN=C2C=N1


InChi: InChI=1S/C18H19ClFN7/c1-27-6-4-11(5-7-27)25-18-21-9-15-16(26-18)17(23-10-22-15)24-12-2-3-14(20)13(19)8-12/h2-3,8-11H,4-7H2,1H3,(H,21,25,26)(H,22,23,24)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥360 days if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.


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