Sodium Channel inhibitor 1

filler

Catalog No. Size 价格库存数量
S3232-2 Solid 2 mg ¥120
售罄
不可用
S3232-10 Solid 10 mg ¥360
售罄
不可用

详情描述

Sodium Channel inhibitor1, one of 3-Oxoisoindoline-1-carboxamides, is a novel and selective voltage-gated sodium channel for pain treatment. IC50 Value: 0.16 uM ( Na v1.7, V hold-90mV); 0.41 uM (Na v1.7, V hold-90mV) Target: Na v1.7Sodium Channel inhibitor1 demonstrated concentration-dependent efficacy in preclinical behavioral pain models.

Product information

CAS Number: 1198117-23-5

Molecular Weight: 473.42

Formula: C24H19F4N3O3

Chemical Name: 7-fluoro-3-oxo-2-[2-(pyridin-2-yl)ethyl]-N-{[4-(trifluoromethoxy)phenyl]methyl}-2,3-dihydro-1H-isoindole-1-carboxamide

Smiles: O=C1C2=CC=CC(F)=C2C(C(=O)NCC2=CC=C(C=C2)OC(F)(F)F)N1CCC1=CC=CC=N1

InChiKey: GRXUKFHZQDPFAI-UHFFFAOYSA-N

InChi: InChI=1S/C24H19F4N3O3/c25-19-6-3-5-18-20(19)21(31(23(18)33)13-11-16-4-1-2-12-29-16)22(32)30-14-15-7-9-17(10-8-15)34-24(26,27)28/h1-10,12,21H,11,13-14H2,(H,30,32)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥360 days if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

相似产品

Recently viewed