详情描述
PFK-015 is a potent inhibitor of PFKFB3. The preliminary results in a U87GM xenograft model have shown that PFK-015 has comparable activity to Temozolomide. PFK-015 inhibits glucoseuptake by tumors.
Product information
CAS Number: 4382-63-2
Molecular Weight: 260.29
Formula: C17H12N2O
Synonym:
PFK015
PFK 015
Chemical Name: (2E)-1-(pyridin-4-yl)-3-(quinolin-2-yl)prop-2-en-1-one
Smiles: O=C(/C=C/C1=CC=C2C=CC=CC2=N1)C1C=CN=CC=1
InChiKey: UJJUKZPBUMCSJZ-BQYQJAHWSA-N
InChi: InChI=1S/C17H12N2O/c20-17(14-9-11-18-12-10-14)8-7-15-6-5-13-3-1-2-4-16(13)19-15/h1-12H/b8-7+
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.