Catalog No. Size 价格库存数量
S2109-2 Solid 2 mg ¥105
S2109-10 Solid 10 mg ¥315


Laropiprant, aslo known as MK-0524, was a drug used in combination with niacin to reduce blood cholesterol (LDL and VLDL) that is no longer sold, due to increases in side-effects with no cardiovascular benefit. Laropiprant itself has no cholesterol lowering effect, but it reduces facial flushes induced by niacin. Laropiprant acts as a selective DP1 antagonist, reducing the vasodilation.

Product information

CAS Number: 571170-77-9

Molecular Weight: 435.90

Formula: C21H19ClFNO4S

Chemical Name: 2-[(3R)-4-[(4-chlorophenyl)methyl]-7-fluoro-5-methanesulfonyl-1H,2H,3H,4H-cyclopenta[b]indol-3-yl]acetic acid

Smiles: CS(=O)(=O)C1=CC(F)=CC2=C1N(CC1C=CC(Cl)=CC=1)C1[C@@H](CC(O)=O)CCC=12


InChi: InChI=1S/C21H19ClFNO4S/c1-29(27,28)18-10-15(23)9-17-16-7-4-13(8-19(25)26)20(16)24(21(17)18)11-12-2-5-14(22)6-3-12/h2-3,5-6,9-10,13H,4,7-8,11H2,1H3,(H,25,26)/t13-/m1/s1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥360 days if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.


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